
Dehydro Nifedipine NEW
Price | $42 | $98 | $147 |
Package | 1mg | 5mg | 10mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2025-05-01 |
Product Details
Product Name: Dehydro Nifedipine | CAS No.: 67035-22-7 |
Purity: 98.65% | Supply Ability: 10g |
Release date: 2025/05/01 |
Product Introduction
Bioactivity
Name | Dehydro Nifedipine |
Description | Dehydro Nifedipine (BAY-b 4759) is the main metabolite of nifedipine in human plasma. Dehydro Nifedipine inhibits glucose uptake in PC-12 cells with an IC50 value of 130 μM. Nifedipine is a calcium channel blocker used in the treatment of hypertension and angina. Dehydronifedipine is formed when it is metabolized by cytochrome P450 (CYP) isomers CYP3A4 and CYP3A5. |
In vitro | Dehydro nifedipine inhibits glucose uptake in PC-12 cells with an IC50 value of 130 μM[1]. |
Storage | store at low temperature | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
Solubility Information | Ethanol : 2.7 mg/mL (7.84 mM), Sonication is recommended. DMSO : 27 mg/mL (78.42 mM), Sonication is recommended. DMF : 30 mg/mL (87.13 mM), Sonication is recommended. DMSO:PBS (pH 7.2) (1:10) : 0.1 mg/mL (0.29 mM), Sonication is recommended. |
Keywords | DrugMetabolite | Drug Metabolite | Dehydro Nifedipine | calcium channel |
Inhibitors Related | Nortriptyline hydrochloride | Clofibric acid | Oseltamivir acid | Mycophenolate Mofetil | Clozapine N-Oxide | Monomethyl fumarate | Monobutyl Phthalate | Isonicotinic acid | Ampyrone | 4-Methylamino antipyrine | Nicotinamide N-oxide | DP-1 hydrochloride |
Related Compound Libraries | Pain-Related Compound Library | Bioactive Compound Library | Membrane Protein-targeted Compound Library | Calcium Channel Compound Library | Anti-Cardiovascular Disease Compound Library | Bioactive Compounds Library Max | Ion Channel Targeted Library | Human Metabolite Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, MA
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