6211-32-1

基本信息
育亨賓堿
洛芙素鹽酸鹽
蘿芙素鹽酸鹽
ALPHA-鹽酸育亨賓
育亨賓提取物 育亨賓堿
蘿芙素鹽酸鹽(甄準(zhǔn)不供應(yīng))
育亨賓鹽酸鹽, 來源于育亨賓
RAUWOLSCINE
ISOYOHIMBINE
MESOYOHIMBINE
RAUWOLSCINE HCL
ALPHA-YOHIMBINE
ALPHA-YOHIMBINE HCL
YOHIMBINE HCL, ALPHA-
RAUWOLSCINE HYDROCHLORIDE
Isoyohimbine hydrochloride
安全數(shù)據(jù)
報價日期 | 產(chǎn)品編號 | 產(chǎn)品名稱 | CAS號 | 包裝 | 價格 |
2025/02/08 | HY-12710 | 育亨賓堿 Rauwolscine | 6211-32-1 | 1 mg | 2320元 |
2025/02/08 | HY-12710 | 育亨賓堿 Rauwolscine | 6211-32-1 | 5 mg | 5800元 |
2025/02/05 | S5337 | 育亨賓堿 Rauwolscine hydrochloride | 6211-32-1 | 25mg | 795.33元 |
常見問題列表
Target | Value |
α2 adrenergic receptor
() | 12 nM(Ki) |
[ 3 H]Rauwolscine binding to α2 adrenergic receptor is reversible, stcreospccific, and saturable. [ 3 H]Rauwolscine specifically labels both the high and low affinity states of the α2 adrenergic receptor in brain membranes. [ 3 H]Rauwolscine also behaves as a 5-HT1A receptor agonist and this conclusion is compatible with earlier functional studies, indicating that rauwolscine (as well as yohimbine) has agonistic properties at the level of 5-HT autoreceptors. When using [ 3 H]5-HT as a radioligand, rauwolscine is determined to have relatively high affinity for the human receptor (K i human=14.3 nM, K i rat=35.8 nM). Saturation studies shows that the affinity of [ 3 H]Rauwolscine is similar in mouse, rat, rabbit, dog (2.33-3.03 nM) except man where it is significantly higher (0.98 nM) .