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216685-07-3

中文名稱 216685-07-3
英文名稱 AR-C117977
CAS 216685-07-3
分子式 C25H28N2O3S2
分子量 468.63
MOL 文件 216685-07-3.mol
216685-07-3 結(jié)構(gòu)式 216685-07-3 結(jié)構(gòu)式

基本信息

英文別名
AR-C117977
AR-C-117977
AR-C 117977
5-((3-hydroxypropyl)thio)-1-isobutyl-3-methyl-6-(naphthalen-1-ylmethyl)thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione
5-(3-hydroxypropylsulfanyl)-3-methyl-1-(2-methylpropyl)-6-(naphthalen-1-ylmethyl)thieno[2,3-d]pyrimidine-2,4-dione
Thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione, 5-[(3-hydroxypropyl)thio]-3-methyl-1-(2-methylpropyl)-6-(1-naphthalenylmethyl)-

應(yīng)用領(lǐng)域

用途一
AR-C117977 is a potent MCT1 inhibitor, which can reduce vimmune responses both in vitro and in vivo, maintains long-term graft survival, and induces operational tolerance.
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