Hazard Information | Back Directory | [Description]
AA10 is a irreversible transglutaminase 2 (TG2) inhibitor. | [Uses]
AA10 is a potent and irreversible transglutaminase 2 (TG2) inhibitor for cancer research[1]. | [References]
[1] Akbar A, et al. Structure-Activity Relationships of Potent, Targeted Covalent Inhibitors That Abolish Both the Transamidation and GTP Binding Activities of Human Tissue Transglutaminase. J Med Chem. 2017 Sep 28;60(18):7910-7927. DOI:10.1021/acs.jmedchem.7b01070 |
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