| Identification | Back Directory | [Name]
Pyrrolo[3,2-c]azepin-4(1H)-one, 5-[3-[4-(4-fluorophenyl)-1-piperazinyl]propyl]-5,6,7,8-tetrahydro-8-hydroxy-1-methyl- | [CAS]
191592-09-3 | [Synonyms]
5-HT2 antagonist 1
Pyrrolo[3,2-c]azepin-4(1H)-one, 5-[3-[4-(4-fluorophenyl)-1-piperazinyl]propyl]-5,6,7,8-tetrahydro-8-hydroxy-1-methyl- | [Molecular Formula]
C22H29FN4O2 | [MDL Number]
MFCD31544447 | [MOL File]
191592-09-3.mol | [Molecular Weight]
400.49 |
| Chemical Properties | Back Directory | [Boiling point ]
613.9±55.0 °C(Predicted) | [density ]
1.28±0.1 g/cm3(Predicted) | [storage temp. ]
Store at -20°C | [solubility ]
Soluble in DMSO | [pka]
14.38±0.20(Predicted) |
| Hazard Information | Back Directory | [Uses]
5-HT2 antagonist 1 is a potent antagonist of 5-HT2 receptor, with weak α1 adrenoceptor blocking activity. | [IC 50]
5-HT2 Receptor; α1 | [storage]
Store at -20°C | [References]
[1] Mizuno A, et al. Synthesis and serotonin 2 (5-HT2) receptor antagonist activity of 5-aminoalkyl-substituted pyrrolo[3,2-c]azepines and related compounds. Chem Pharm Bull (Tokyo). 2000 May;48(5):623-35. DOI:10.1248/cpb.48.623 |
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