| Identification | Back Directory | [Name]
Ethanone, 1-[3-(5-methoxy-1H-indol-3-yl)-1-piperidinyl]- | [CAS]
190328-44-0 | [Synonyms]
GR128107
GR-128107
GR 128107
Ethanone, 1-[3-(5-methoxy-1H-indol-3-yl)-1-piperidinyl]- | [Molecular Formula]
C16H20N2O2 | [MOL File]
190328-44-0.mol | [Molecular Weight]
272.34 |
| Hazard Information | Back Directory | [Description]
GR 128107 is a melatonin receptor antagonist. | [Uses]
GR 128107 is a competitive melatonin receptor antagonist (pKi: 9.6)[1]. | [References]
[1] Dubocovich ML, et al. Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75. DOI:10.1007/pl00004956 |
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